Highly Substituted Isoxazoles: The Baylis-Hillman reaction of substituted 4-isoxazolecarbaldehydes and attempted cyclization to isoxazole-annulated derivatives
IR@CDRI: CSIR-Central Drug Research Institute, Lucknow
View Archive Info| Field | Value | |
| Creator |
Roy, Amrendra K
Batra, Sanjay |
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| Date |
2007-11-15T05:42:40Z
2007-11-15T05:42:40Z 2003 |
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| Identifier |
Synthesis (2003)1347-1356
http://hdl.handle.net/123456789/20 |
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| Description |
In an attempt to understand the effect of position of the formyl group on the efficiency of Baylis-Hillman reaction within isoxazolecarboxaldehydes, the reactions of substituted 4-isoxazolecarboxaldehydes to obtain highly substituted isoxazoles are described. Attempts to obtain isoxazole-annealed derivatives from these Baylis-Hillman adducts involving SNR’-SNAr substitu-tion strategy are also described.
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| Format |
141205 bytes
application/pdf |
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| Language |
en
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| Relation |
CDRI Communication Number 6389
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| Subject |
Baylis-Hillman reaction
DABCO DMAP. 4-isoxazolecarboxaldehyde |
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| Title |
Highly Substituted Isoxazoles: The Baylis-Hillman reaction of substituted 4-isoxazolecarbaldehydes and attempted cyclization to isoxazole-annulated derivatives
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| Type |
Article
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